Galantamine Hydrobromide powder olupese CAS No.: 1953-04-4 98% mimo min.fun awọn eroja afikun
Ọja paramita
Orukọ ọja | Galantamine Hydrobromide |
Oruko miiran | Galanthamine hydrobromide; Galantamine HBr; Galanthamine HBr; (4aS,6R,8aS) -4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-6H-Benzofuro [3a,3,2-ef] [2] benzazepin- 6-ol, Hydrobromide |
CAS No. | Ọdun 1953-04-4 |
Ilana molikula | C17H21NO3.HBr |
Ìwúwo molikula | 368.27 |
Mimo | 98.0% |
Ifarahan | funfun si pa-funfun lulú |
Iṣakojọpọ | 1kg/apo 10kgs ,25kgs / ilu |
Ohun elo | nootropics |
ifihan ọja
Galantamine hydrobromide jẹ iru benzozepine ti o wa lati awọn isusu ati awọn ododo ti narcissus, osmanthus, tabi canna.O tun jẹ onidalẹkun cholinesterase oral.Gẹgẹbi ligand ti nicotinic acetylcholine receptor, o ti ni lilo pupọ lati mu iṣẹ neurocognitive ṣiṣẹ.Ipa rẹ ni lati ni ifigagbaga ati ni iyipada ni idiwọ acetylcholinesterase, nitorinaa jijẹ ifọkansi ti acetylcholine.
Nigbati o ba wọ inu ẹjẹ, galanthamine hydrobromide ti wa ni irọrun gba sinu gbogbo awọn ẹya ara, pẹlu ọpọlọ.O sopọ mọ olugba acetylcholine nicotinic, nfa awọn iyipada isọdi ati jijẹ itusilẹ acetylcholine.O tun ṣiṣẹ nipasẹ idije ati yiyipada awọn ipa ti awọn inhibitors cholinesterase.Nipa idinamọ cholinesterase, o ṣe idiwọ jijẹ ti acetylcholine, nitorina o pọ si ipele ati iye akoko ti neurotransmitter ti o lagbara yii.Galanthamine tun ṣe ilọsiwaju ẹkọ ati agbara iranti, ṣe idiwọ iredodo ọpọlọ ati ṣetọju awọn ipele giga ti awọn neurotransmitters nipa mimu iduroṣinṣin ti awọn neuronu ati awọn synapses.
Ẹya ara ẹrọ
(1) Ipa miiran ti o niyelori ti galanthamine hydrobromide lori imudara iranti ni agbara rẹ lati mu iṣẹ iranti pọ si.O mu iyara ti idasile iranti pọ si ati ilọsiwaju idaduro awọn alaye ati awọn otitọ.
(2) Agbara ikẹkọ ti ni ilọsiwaju nipasẹ jijẹ ṣiṣu synapti ati neuroplasticity.Galanthamine hydrobromide taara tabi aiṣe-taara ni ipa lori neuroplasticity.O nmu pilasitik synapti ṣiṣẹ nipasẹ mimuuṣiṣẹpọ microglia ati astrocyte.
(3) O ṣe iranlọwọ fun oorun ati mu isinmi pọ si.Galanthamine le mu iṣoro ti iṣẹlẹ oorun pọ si nipa ti nfa oorun gbigbe oju iyara ni kutukutu, nitorinaa imudarasi didara oorun.
(4) Ṣe ilọsiwaju idaabobo ẹda, Galantamine n pese idaabobo ẹda lati koju aapọn oxidative ti o ṣẹlẹ nipasẹ awọn ipilẹṣẹ ọfẹ.O le daabobo awọn sẹẹli ọpọlọ lati ibajẹ oxidative lati ṣetọju iṣẹ ọpọlọ ti o dara julọ.