Nefiracetam powder olupese CAS No.: 77191-36-7 99% mimo min.fun awọn eroja afikun
Ọja paramita
| Orukọ ọja | Nefiracetam |
| Oruko miiran | n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamide; NEFIRACETAM; 2-oxo-1-pyrrolidinylaceticacid,2,6-dimethylanilide; dm9384; n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamid; DM-9384, (2- (2-Oxopyrrolidin-1-yl) -N- (2,6-dimethylphenyl) -acetamide; DMMPA |
| CAS No. | 77191-36-7 |
| Ilana molikula | C14H18N2O2 |
| Ìwúwo molikula | 246.3 |
| Mimo | 99.0% |
| Ifarahan | Iyẹfun funfun |
| Iṣakojọpọ | 25 kg / agba |
| Ohun elo | nootropic |
ifihan ọja
Nefiracetam je ti si awọn ti kii-aala itetisi kilasi imudara kilasi ti oloro, eyi ti o ni orisirisi awọn kemikali ẹya ati ki o mu imo agbara ati ki o se awọn bibajẹ ti eko ati iranti nipasẹ wọn ipa lori cerebral kotesi.Ko ni awọn ohun-ini ti muscarinic receptor agonists ati antagonists, tabi ko ṣe idiwọ iṣẹ ṣiṣe ti Ach.Awọn ipakokoro-igbagbe ati awọn igbelaruge iranti ti oogun yii jẹ aṣeyọri nipasẹ imudara itusilẹ ti Ach ni kotesi cerebral.Awọn kinases amuaradagba ti o gbẹkẹle ibudó ṣe alekun iṣẹ ṣiṣe ikanni Ca2+, eyiti o le jẹ iduro fun itusilẹ Ach wọn ti mu dara si.Nefiracetam (NEF) jẹ aṣoju nootropic iru pyrrolidone pẹlu ọpọlọpọ awọn oogun oogun bii awọn ipa imudara imọ.Ni amygdala-kindled imulojiji, nefiracetam dojuti mejeeji electroencephalographic ati ihuwasi imulojiji.NEF ni a pato anticonvulsant julọ.Oniranran.
Ẹya ara ẹrọ
Nefiracetam ti wa ni lo lati toju cerebrovascular arun.O le mu agbara oye pọ si ati ṣe idiwọ ibajẹ ti ẹkọ ati iranti nipasẹ ipa rẹ lori kotesi cerebral.Ko ni awọn ohun-ini ti agonist olugba muscarinic ati oluranlowo antagonistic, tabi ko ṣe idiwọ iṣẹ ṣiṣe ti acetyl cholinase.Nitorina, egboogi-igbagbe ati awọn ipa imudara iranti waye nipasẹ imudarasi itusilẹ ti acetylcholine ni kotesi cerebral.
Awọn ohun elo
Nefiracetam jẹ itọsẹ hydrophobic ti piracetam ati iṣelọpọ sintetiki ti gbogbo awọn agbo ogun Racetam piracetam.Nefiracetam ti ṣelọpọ nipataki nipasẹ Daiichi Sankyo (ile-iṣẹ elegbogi Japanese) fun itọju AD.Ni afikun si gbogbo awọn ọna ṣiṣe ti a sọ si Nefiracetam, o jẹ ero gbogbogbo pe o jẹ nkan ti o ni iduro fun wiwa awọn ikanni kalisiomu ninu ara, ati gbigbe aiṣe-taara ti nkan isamisi ayọ, ti n ṣiṣẹ bi agonist apakan ti glycine-abuda aaye ti olugba NDMA.
